Clenbuterol

Description overdue on 11/15/2014

• Latin name: Clenbuterol
• ATC code: R03CC13
• Active substance: Clenbuterol (Clenbuterol)
• Manufacturer: Balkan Pharmaceuticals UK Ltd, Moldova

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• Composition
• Product form
• Pharmacological action
• Pharmacodynamics and pharmacokinetics
• Indications
• Contraindications
• Side effects
• Clenbuterol syrup, instructions for use (method and dosage)
• Overdose
• Cooperation
• Terms of sale
• Storage conditions
• Shelf life
• Cautions
• Analogs
• Babies
• With alcohol
• Slimming
• During pregnancy (and lactation)
• Reviews
• Price, where to buy

Composition

1 ml of the syrup composition includes the following components:

• clenbuterol hydrochloride   - 1 g;
• sorbitol - 280 mg;
• Glycerol - 200 mg;
• propylene glycol - 100 mg;
• citric acid monohydrate - 7 mg;
• Sodium citrate dihydrate - 5, 8 mg;
• ethanol solution with a concentration of 96% - 5 mg;
• methyl parahydroxybenzoate - 0, 45 mg;
• Propyl - 0, 05 mg;
• butilparagidroksibenzoat - 0, 05 mg;
• sodium benzoate - 1, 2 mg;
• raspberry liquid form - 0, 45 mg;
• Purified water to 1 ml.

Product form

• The pharmacy Clenbuterol from company sold the Balkans as a clear, slightly viscous Syrup Which has a light yellow color with a characteristic smell of raspberry. This form is packaged in drug vials are of dark glass (or dark terephthalate) in 100 ml. Carton contains 1 bottle with a pharmaceutical preparation, measuring cup and spoon set.
• You can also find the company's products in the form Vermodzhe tablets tradename Clenbuterol Ver. But this form of the pharmaceutical agent is not gained wide popularity due to unreasonably high prices.

Pharmacological action

Clenbuterol - active drug, which is based on the eponymous selective beta2-agonists   - Biological active component stimulating corresponding receptors of the human body, preferably located in the bronchial tree of the respiratory system.

Mechanism of action   Biochemical not very complex, it can be represented as a series of sequential reactions. In response, the local penetration of the components of the pharmaceutical formulation into the lumen of the bronchi activated cycle secondary messengers : Adenylyl cyclase - cAMP - Protinkinaza A. Next Clenbuterol influence extend to the myosin, which is localized in the smooth muscle fibers that interact with actin leads to a relaxation of the bronchi. Thus docked abnormal narrowing of the breathing tube during attacks of asthma or chronic obstructive pulmonary disease.

Clenbuterol also affect secretory feature respiratory system. As is known, the reaction of inflammation or other pathological mechanisms are closely related to the allocation of appropriate biological mediators or other active agents that promote bronchoconstriction. The therapeutic effect of the drug slows their release, which is manifested in the elimination of stagnation, reduce edema and normalization mucociliary clearance .

Note that Clenbuterol used in sports medicine In particular the widespread use of a pharmaceutical formulation found in bodybuilders. Active drug ingredients have anabolic effect   Like natural or artificial steroids However they exhibit with a smaller force. Because cough syrup can be used as a fat burner when drying in order to increase the relief of muscular body. The visual effects of the use of a pharmaceutical formulation compared with an incredibly long low-calorie diet.

Pharmacodynamics and pharmacokinetics

The drug is used enterally Then completely absorbed from the digestive tube. Clenbuterol begins to act 10-15 minutes after oral administration, and the maximum therapeutic properties manifest themselves in 2-3 hours. Metabolized active ingredients of the pharmaceutical formulation in the liver. 78 percent of metabolites excreted in the urine. The remainder of the metabolites is eliminated with bile into the lumen of the gastrointestinal tract.

Indications

• bronchial asthma ;
• chronic obstructive pulmonary disease.

Contraindications

• increased individual sensitivity to the constituent components of the drug;
• tachycardia   and tachyarrhythmia;
• severe coronary artery disease;
• thyrotoxicosis ;
• acquired or hereditary intolerance biologically active substances Clenbuterol;
• idiopathic hypertrophic subaortic stenosis of the aorta;
• acute phase myocardial infarction .

Also, the appointment of a pharmaceutical preparation should consider not absolute contraindications, the presence of which recommended a course of conservative therapy in rehabilitation departments under the supervision of medical personnel and must conduct clinical trials:

• diabetes ;
• chronic ischemic heart disease;
• hyperthyroidism ;
• expressed arterial hypertension ;
• cardiomyopathy;
• the presence or susceptibility to arrhythmias ;
• heart defects:
• other dangerous diseases of the cardiovascular system.

Side effects Clenbuterol

Side effects of pharmaceutical formulation affect many organs and systems, as after the absorption of active ingredients carried by the main blood flow. There may be:

• On the part of the cardiovascular system - tachycardia and other kinds of heart palpitations up to the subjective sensations, increased Blood Pressure , Arrythmia, pain in the heart muscle.
• From the nervous system - headache   dizziness, anxiety, insomnia and other sleep disorders, tremor   fingers with deliberate motor act (for example, during the finger-nose test).
• Gastrointestinal tract - dry oral spilled abdominal pain . nausea and following vomiting.
• Local and generalized allergic reactions - hives , Skin rash, acute localized angioedema , Abnormal transient narrowing of the bronchial lumen.
• From the other systems of organs and tissues - muscle spasms   and cramps, intense flow of blood to the face (clearly visible pink cheeks), increased sweating, hypokalemia, and, as a consequence, muscle pain, patients characterized as "body aches."

Of special note is the development of muscle cramps   when using Clenbuterol bodybuilders, since the dosage of the pharmaceutical preparation in the sport is much higher than therapeutic. This side effect is caused by depletion of endogenous reserves Taurine , Deficiency of electrolytes sodium and potassium, with a total lack of water-salt metabolism. To relieve muscle spasms recommended the following changes in the diet:

• use copious amounts of fruit (particularly bananas, since they contain a lot of potassium);
• excessive drinking;
• additional incorporation of taurine in an amount of 3-5 grams per day;
• potassium supplements tablet daily at bedtime on an empty stomach (at least 200-400 mg).

Clenbuterol syrup, instructions for use (method and dosage)

Instructions for clenbuterol for therapeutic purposes

Syrup for use enterally inwardly. Optimal dosage category for adult patients of 15 ml 2-3 times a day in the early conservative therapy of pharmaceuticals. Further, after the elimination of the major symptoms of asthma or chronic obstructive lung disease, supports the applied dosage of 10 ml, 2 times a day.

Duration conservative rehabilitation is 8-10 weeks, but the drug should be taken under the special scheme since anabolic properties of existing components. The course consists of 2 weeks of continuous reception and 2 weeks of "rest" when the syrup is not used alternately, until the attending physician deems it necessary to stop further use of the syrup.

Clenbuterol can be used in pediatric practice. Dosage for children It depends on age and body weight, and makes the following figures:

• children up to 8 months, with a mass of 4.8 kg - 2, 5 ml 2 times a day;
• from 8 months to 2 years old (weighing about 8-12 kg) - 5 ml, 2 times a day;
• the age group of 2 to 4 years of age (12-16 kg) - 7, 5 ml, 2 times a day;
• children of 4 to 6 years of age and weighing 16-22 kg under - 10 ml, 2 times a day;
• from 6 to 12 years (22-35 kg) - 15 ml 2 times a day;
• children over 12 years weighing more than 35 kg - 15 ml 2-3 times a day.

Instructions for use in bodybuilding

Drying Body   - Slang expression, which recently used not only in professional sports and bodybuilding, but also ubiquitous in gyms or youth. Sportswiki It explains this neologism as getting rid of the subcutaneous fat, to give the body "carved" muscle relief. The ultimate goal of drying is dry, smart appearance, and not just getting rid of the extra kilos.

In order to achieve the desired results, in addition to physical exercise can be used: Sports nutrition   or Pharmaceutical preparations Accelerating metabolism and metabolic processes incorporating more fat than normal. So, for example, clenbuterol sportviki and other related sites is as firm as the optimal drug with a short list of possible side effects and is well marked positive effect on the athlete's body.

Course Clenbuterol drying

The dosage of the pharmaceutical preparation contains in micrograms, which corresponds to the dry residue of the active ingredients of syrup to be calculated independently or with the assistance of qualified professionals. It is strictly forbidden to equate the weight and bulk of the drug.

Driving, drinking Clenbuterol for drying:

• 1 day - 20 mg;
• Day 2 - 40 g;
• Day 3 - 60 mg;
• Day 4 - 80 mg;
• Day 5 - 100 g;
• 6-12 days - 120 mg;
• Day 13 - 80 g;
• Day 14 - 40 micrograms.

Next, you need to do, at least, two-week break   before going through the next course of treatment with a pharmaceutical preparation. The optimal time for the reception syrup drying   morning As well as the absorptive capacity of higher organisms. Moreover, thus avoiding the possible development of insomnia.

How to increase the effectiveness of the course

Clenbuterol - a strong anabolic pharmaceutical preparation, but for the development of the effects noticeable to the naked eye it requires a certain amount of time. Depending on the individual sensitivity may take several courses drying. Because experienced athletes, bodybuilders   I recommend taking it along with some other drugs and elements of sports nutrition. First muscle definition will be evident much earlier in this case, on the other hand - there are pharmaceutical preparations that minimize the risk of side effects.

For example, drying can be presented as a course of Clenbuterol + Yohimbine + Ketotifen. The first component is used on the basis of its anabolic effects, ie directly to satisfy the desire to spend the subcutaneous fat and achieve the desired shape and muscle relief. Why use Ketotifen   described below. Yohimbine In turn, it is a plant alkaloid with a pronounced stimulating action. For therapeutic purposes it is used as aphrodisiac recovery of erectile dysfunction. Bodybuilders Yohimbine is used to increase the effect of anabolic steroids and prevention of genital problems.

How to take Clenbuterol and Ketotifen

Ketotifen - pharmaceutical drug that is often used in bodybuilding. Its active ingredients have almost unique therapeutic properties - they allow restore sensitivity andrenoretseptorov   to drugs and anabolic clenbuterol in particular. This ability of the drug more than once proved in clinical trials. With Ketotifenum can be 10-20 percent increase efficiency   conservative course and greatly accelerate the process of drying or weight loss. Another positive feature of the drug is possible to compensate for such adverse effects as mental stimulation, rhythm disorders of sleep and wakefulness, and some others.

The recommended course of Clenbuterol and ketotifen on drying:

• 1 day - 20 mg Clenbuterol;
• Day 2 - 40 mcg Clenbuterol;
• Day 3 - 60 mcg Clenbuterol;
• Day 4 - 80 mcg Clenbuterol;
• Day 5 - 100 mcg of Clenbuterol and 1 mg ketotifen;
• 6-27 days - 120 mcg of Clenbuterol and 2 mg ketotifen;
• Day 28 - 80 mcg Clenbuterol and 2 mg ketotifen;
• Day 29 - 50 mcg Clenbuterol ketotifen and 1-2 mg, depending on the subjective sensation;
• Day 30 - 33-35 mcg Clenbuterol and 1 mg ketotifen.

Preferably use Clenbuterol in the morning, and Ketotifen - at night, before bedtime. Break before the next course of use of pharmaceuticals should be at least two weeks.

How to take Clenbuterol + Yohimbine + Thyroxine

The high efficiency of the complex due to the inclusion in it Thyroxine   - this thyroid hormone Which is produced normally in a healthy body. For drying, it is used for two reasons - first of all an active thyroxine physiological fat burner Capable of self-accelerating metabolism and launch relevant metabolic processes. Second, its effects extend to the adrenergic receptors, which act through Clenbuterol and Yohimbine, ie indirectly Thyroxine enhances the effect of other fat burners metabolism. Thus, to create an optimal biochemical environment for the rapid disposal of unnecessary kilograms.

1 operating unit of the complex is:

• Clenbuterol 40 mg (syrup should be recalculated on the dry residue);
• Thyroxine - 25 g;
• Yohimbine - 5 mg.

The recommended course of taking must comply with the following scheme:

• 1-3 day - 1 unit;
• 4-6 day - 1, 5 units;
• 7-9 day - 1 unit 1 unit in the morning and afternoon;
• 10-12 days - 1, 5 units;
• Day 13-15 - 1 unit;
• Day 16-19 - 0, 5 units;
• 20-21 days - 0, 25 units.

This is followed by a break of at least 3-4 weeks, and you can repeat the course under the same scheme. Take pharmaceuticals recommended 30 minutes before breakfast, with a small amount of ordinary drinking water.

With the development of side effects Such as fever, should consult a doctor or trainer. You also need to implement prophylactic 1-2 mg Ketotifenum after noon. To avoid possible problems with the heart and reduce the incidence of myocardial contractions necessary to use beta-blockers - Metoprolol   50 mg 2 times a day.

Clenbuterol is prohibited or not in sports?

In addition to the external effects associated with a decrease in body fat, a pharmaceutical formulation enhances the body's performance and to some extent increase the power rates. Since 1992 Anti-Doping Committee banned the use of the drug by professional athletes. However, bodybuilders at the amateur level Clenbuterol remains popular and still, as its effects are clearly visible after passing the respective course.

Overdose

Be sure to consult how to take Clenbuterol for drying, slimming or therapeutic purposes in the presence of an active pathological process with the respective qualified personnel or pharmacists, because the drug can cause an overdose condition, characterized by the following symptoms:

• heart palpitations ;
• cardiac arrhythmias;
• hypokalemia;
• hypertension (up to hypertensive crises);
• kardialgiya;
• trembling of the upper and lower extremities.

Pharmaceutical antidote for Clenbuterol is not because an overdose of a drug used symptomatic and detoxification therapy. First of all, if the above symptoms occur, you should clean the upper gastrointestinal tract of active chemical components in all possible ways (gastric lavage, oral adsorbents, and so on). Further, to restore the disturbed metabolic properties of the body, which are generally used water and brine. Well, it is imperative in overdose contact your doctor.

Cooperation

The drug has a very broad list of clinical interaction, which is required to be taken into account when Clenbuterol is used for drying or for therapeutic purposes:

• in combination with monoamine oxidase inhibitors   (MAO) and Theophylline violates conduction of impulses to the heart muscle;
• antagonism (the opposite direction of action) with beta-blockers ;
• It raises the possibility of arrhythmic condition at admission cardiac glycosides ;
• hypoglycemics   loses much of its therapeutic efficacy, respectively, an increase in dosage is required at the time of the course Clenbuterol;
• in combination with simpatomimetikami increases the toxicity of the active ingredients of the pharmaceutical formulation.

Terms of sale

Buy Clenbuterol syrup can only be certified by the attending physician for a prescription.

Storage conditions

Keep a pharmaceutical formulation should be protected from light, with a moderate regime of humidity and temperatures above 25 degrees Celsius. Also dosage pills should be out of reach of young children place.

Shelf life

3 years.

Cautions

Match code ATC 4th level:

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Babies

During pregnancy and lactation

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