Clenbuterol Sopharma

Description overdue on 10/17/2014

• Latin name: Clenbuterol Sopharma
• ATC code: R03CC13
• Active substance: Clenbuterol Hydrochloride (Clenbuteroli hydrochloridi)
• Manufacturer: "Sopharma" JSC Bulgaria («Sopharma» AD (Bulgaria)

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• Composition
• Product form
• Pharmacological action
• Pharmacodynamics and pharmacokinetics
• Indications
• Contraindications
• Side effects
• Clenbuterol tablets, instructions for use (method and dosage)
• Overdose
• Cooperation
• Terms of sale
• Storage conditions
• Shelf life
• Cautions
• Babies
• Slimming
• During pregnancy (and lactation)
• Reviews
• Price, where to buy

Composition

1 tablet pharmaceutical drug Clenbuterol Sopharma includes such components as:

• Clenbuterol Hydrochloride   (primary active agent) - 0, 2 mg;
• lactose monohydrate - 70 mg;
• microcrystalline cellulose (MCC) - 48, 5 mg;
• Wheat starch - 31, 48 mg;
• Povidone K 25 - 6 mg;
• colloidal silica - 2 mg;
• magnesium stearate - 2 mg.

1 ml Syrup in its composition has the following components:

• Clenbuterol Hydrochloride - 1 g;
• sorbitol;
• glycerol;
• propylene glycol;
• sodium citrate;
• citric acid monohydrate;
• methyl parahydroxybenzoate, propyl parahydroxybenzoate and butilparagidroksibenzoat;
• sodium benzoate;
• essence "Raspberry" in liquid form;
• purified water.

Product form

Pharmacies medicament can be found in the form:

• Tablets Klenbutrol   at 0, 2 mg each. Packed in blisters (blisters of aluminum foil or PVC) of 10 pieces. Cardboard boxes can hold, usually 5 plates.
• Transparent and slightly viscous Clenbuterol syrup   colorless to pale yellow with a characteristic smell of raspberry. Packed this form of the drug in vials of dark glass (or dark PET) 100 ml with measured glass and spoon set. Carton contains 1 vial of the pharmaceutical and the above mentioned items.

Pharmacological action

The main component of the drug Clenbuterol Sopharma - a selective beta2-agonists That is, the mechanism of action of the active component comprises a stimulating effect on the type of receptors which are mainly located in bronchial tree . In response to the next activated cycle of secondary messengers   in the following sequence: adenylyl cyclase - cAMP - Protinkinaza A. Then apply to the effect of Clenbuterol myosin Component of smooth muscle fibers which interact with actin, resulting in   relaxation of bronchi . Thus, the problem is eliminated narrowing of the lumen of the respiratory tract during asthma attacks and largely facilitated respiratory processes.

Clenbuterol has and sekretoliticheskim action . In particular, the main component of the pharmaceutical formulation slows the release of inflammatory mediators and other biological active substances from mast cells, which enhance bronchospasm. Thanks to these therapeutic properties decreases swelling , Eliminated the stagnation in the lumen of the bronchial tree, improves mucociliary clearance .

Of special note properties Clenbuterol used in sports pharmacology . The active component of the drug has anabolic properties similar to steroids, but exert their effects with a smaller force. The pharmaceutical preparation is active fat burner . The mechanism of this action is to a slight increase in the internal temperature of the body, thereby increasing the consumption of calories. Among athletes and bodybuilders are of the opinion that the increase in temperature of 1 degree Celsius accelerates the metabolism of fat by 5 percent.

Thanks to these therapeutic effects stiffness muscular frame   and strength far exceeds initial testimony to the passage of the conservative course. The body is attached relief , Vascularity and desired look. Externally, these effects are comparable with prolonged low-calorie diet.

Pharmacodynamics and pharmacokinetics

The drug is used orally Then adequately and well absorbed from the gastrointestinal tract. Clenbuterol begins to act within 10-15 minutes after ingestion, and the maximum therapeutic properties manifest themselves in 2-3 hours. Metabolized the active components of a pharmaceutical preparation in the liver, after which 78 percent of the products of metabolism output urine. A small number of metabolites is eliminated with bile into the lumen of the digestive tube.

Indications

• Bronchial asthma;
• Chronic obstructive pulmonary disease.

Contraindications

• increased individual sensitivity to the constituent components of the drug;
• acquired or hereditary intolerance biologically active substances Clenbuterol Sopharma;
• tachycardia and   tachyarrhythmia;
• thyrotoxicosis ;
• idiopathic hypertrophic subaortic stenosis   aorta;
• severe coronary heart disease ;
• acute phase myocardial infarction .

Conservative treatment Klenbutrolom against the backdrop of these pathologies should be   carefully Which involves treatment in special hospital under constant supervision of qualified medical personnel and regular diagnostic tests:

• hyperthyroidism;
• diabetes ;
• diseases of the cardiovascular system (particularly pronounced hypertension, cardiomyopathy, valvular heart disease, coronary artery disease   or a tendency to arrhythmias ).

Side effects

• From the nervous system - headache   and g olovokruzhenie , Anxiety, disturbance of sleep and wakefulness in the form insomnia , Intention tremor   fingers.
• Cardio-vascular system - tachycardia, increased blood pressure, arrythmia , Kardialgiya.
• Gastrointestinal tract - dryness in the oral cavity, stomachalgia . nausea Resulting in vomiting.
• Local and generalized allergic reactions - hives , Skin rash, bronchospasm, angioedema .
• On the part of other organ systems and tissues - muscle cramps, intense flushing of the face , Increased sweating, hypokalemia and, as a consequence, muscle pain.
• There is a possibility of syndrome "ricochet"   Cancelled and resistance in the pharmaceutical preparation.

Of special note is the development of muscle cramps When Klenbutrol tablets used by athletes and bodybuilders. This side effect is caused by the depletion of stocks of endogenous taurine deficiency of electrolytes sodium and potassium, with a total lack of water-salt metabolism. To relieve muscle spasms recommended The following changes in diet:

• use copious amounts of fruit (particularly bananas, since they contain a lot of potassium);
• excessive drinking;
• additional incorporation of taurine in an amount of 3-5 grams per day;
• potassium supplements tablet daily at bedtime on an empty stomach (at least 200-400 mg).

Clenbuterol tablets, instructions for use (method and dosage)

Syrup indicated for oral administration. For adults   The optimum dosage is 15 ml 2-3 times a day at the beginning of a course of conservative treatment. After arresting the serious condition of the prescribed amount of drug to be reduced to a maintenance dose of 10 ml, 2 times per day.

Instructions on the use of a pharmaceutical formulation and its use permits in pediatric patients But with strict observance of the following dosages:

• children up to 8 months, with a mass of 4.8 kg - 2, 5 ml 2 times a day;
• from 8 months to 2 years old (weighing about 8-12 kg) - 5 ml, 2 times a day;
• the age group of 2 to 4 years of age (12-16 kg) - 7, 5 ml, 2 times a day;
• children of 4 to 6 years of age and weighing 16-22 kg under - 10 ml, 2 times a day;
• from 6 to 12 years (22-35 kg) - 15 ml 2 times a day;
• children over 12 years weighing more than 35 kg - 15 ml 2-3 times a day.

Pills As a syrup, it is administered orally. Dosage pharmaceutical preparation depends on the weight and response of the organism in the form of side effects or adverse effects of the drug. The average amount of the drug for men is around 100-140 mg, and women - 80-100 micrograms per day. Acceptance must start with optimal dosage And accumulate it gradually to provide the maximum therapeutic effect. That is a conservative course starts with 1 tablet per day and then increased by 1 tablet every day.

Duration such treatment is on average about 8-10 weeks. However, a special use regimen medicament as Clenbuterol has not its anabolic effects after 18 days of continuous use. Therefore the course consists of 2 weeks of continuous reception and 2 weeks off alternately until the pharmaceutical preparation will not end or the attending physician does not stop its further use.

Overdose

Admission dosages, highly exceeding the prescribed, accompanied by:

• arrhythmia;
• tachycardia;
• gipolkaliemiey ;
• hypertension;
• tremor limb;
• pain in my heart.

Specific antidote for Clenbuterol not, because as a treatment used detoxification and symptomatic therapy Ie gastric lavage, administration of oral sorbents (for example, Activated Carbon ), The use of aqueous salt solutions to recover the relevant metabolic disorders, monitoring of potassium level in the blood serum and correction of it properly.

Cooperation

In the appointment of Clenbuterol Sopharma, consider the following clinical interaction pharmaceutical formulation:

• antagonism with opposite effects on beta-blockers ;
• violation of intracardiac conduction in the combined use with MAO inhibitors   (monoamine oxidase) and Theophylline ;
• reduction in the efficiency of hypoglycemic agents (requires recalculation of dosages for patients with diabetes);
• increased toxicity   cardiac glycosides (greatly increased risk of developing a pathological condition such as arrhythmia);
• increase the toxicity in combination with   mimetic sympathetic character .

Terms of sale

Dispense medication strictly on prescription, the print confirmation of the attending physician.

Storage conditions

Keep a pharmaceutical formulation should be protected from light, with a moderate regime of humidity and temperatures above 25 degrees Celsius. Also dosage pills should be out of reach of young children place.

Shelf life

3 years

Cautions

The adverse effects of medical treatment pharmaceutical preparations include intentsionnogo tremor . dizziness, weakness , Because during the passage of the therapeutic course should be abandoned   on the performance of potentially hazardous activities that require maximum concentration and speed of reaction. For example, you should not drive a car or other means of transportation.

Babies

The medicament may be used in pediatric practice only on the basis of the above dosages calculated to certain ages and body weight of the child.

Slimming

The medicament may be used as a fat burner in sports pharmacology, as active components increases the internal temperature of the organism (see. Explanation of the mechanism of action above).

During pregnancy (and lactation)

Clenbuterol tablets has, to some extent tocolytic property , because should not   appoint a pharmaceutical product while carrying a child in the prenatal and birth periods. Absolutely contraindicated drug in 1 trimester of pregnancy.

Clinical studies have not reliably confirmed nor denied the fact that the active component is capable of acting passes into breast milk. The lack of relevant data as possible assignment of a pharmaceutical preparation only if the expected utility of the therapeutic effect of the tablets will be largely outweighs the potential risk to the child.

Reviews of Clenbuterol Sopharma

First of all, it should be noted that more feedback on the pharmaceutical preparation, as a means to effectively arrest the spasm of the bronchial tree during attacks asthma . Such therapeutic effect abundantly used in medicine and clinical studies have confirmed the qualified experts. Of course, the drug has certain side effects, but the effect it develops within 10-15 minutes after ingestion, which allows you to quickly eliminate life-threatening pathological condition.

However, discussion forums and online resources found on other reviews and the scope of Clenbuterol. Athletes and bodybuilders prefer to use the pharmaceutical preparation as diet pills   or so-called "drying." This task, as well as the liquidation of the bronchospasm drug copes with a bang, as the basis for such actions are justifiable mechanisms. However, the course is accompanied by severe side effects   in the form of muscle cramps, because, as a rule, these patients seek as soon as possible to lose weight.

We can say that during the course of a conservative administration of the drug Clenbuterol Sopharma should strictly adhere to these instructions dosages. Through such simple actions can save yourself from unnecessary suffering, trips to doctors and other adverse effects.

Price Clenbuterol Sopharma, where to buy

Price Clenbuterol tablets in Ukraine 95 hryvnia for a pharmaceutical formulation in the form of syrup, and 190 hryvnia per tablet. Buy drug may be in the territory of the Russian Federation. So, buy Clenbuterol tablets can be in Moscow for 250 rubles. Cost syrup in Russian pharmacies identical release tablet form drugs.

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